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#7
Le modafinil est souvent utilisГ© Г  titre prГ©ventif pour retarder la somnolence diurne, bien qu'il ait une trГЁs faible chance de devenir une dГ©pendance. Les chercheurs qui ont menГ© l'Г©tude pensent que ces rГ©sultats reprГ©sentent un test du stimulant sur les centres Г©motionnels du cerveau. Ces deux derniГЁres rГ©gions du cerveau sont importantes pour la rГ©gulation du sommeil. Le modafinil a Г©tГ© utilisГ© hors indication pour d'autres troubles du sommeil et de l'Г©veil diurne, tels que le somnambulisme et les troubles du rythme circadien. L'ingrГ©dient modafinil est un dГ©rivГ© de l'amphГ©tamine. Son mГ©canisme d'action est similaire Г  celui de l'amphГ©tamine ; il amГ©liore l'Г©veil et augmente la vigilance. Le modafinil a Г©tГ© dГ©veloppГ© Г  l'origine comme agent favorisant l'Г©veil, mais s'est rГ©vГ©lГ© efficace dans le traitement de diverses autres affections pouvant entraГ®ner une somnolence diurne excessive, notamment les troubles du sommeil liГ©s au travail postГ©, la narcolepsie et certains troubles neurologiques. La dose quotidienne maximale recommandГ©e est de 600 mg. Un mГ©dicament modafinil est un somnifГЁre liГ© aux amphГ©tamines telles que l'amphГ©tamine. Le modafinil peut Г©galement aider les personnes souffrant d'apnГ©e obstructive du sommeil. Ces substances sont normalement fabriquГ©es pendant les pГ©riodes d'Г©veil, la production augmentant dans les heures prГ©cГ©dant l'endormissement. modiodal drogue La Food and Drug Administration (FDA) a approuvГ© ce mГ©dicament pour le traitement de la narcolepsie, des troubles du sommeil liГ©s au travail postГ© et de l'apnГ©e obstructive du sommeil. L'adГ©nosine est responsable de la production de sommeil dans le cerveau. Bien qu'il porte de nombreux surnoms, notamment Nuvigil, Armodafinil et Provigil, le mГ©dicament est Г©galement connu simplement sous le nom de M100. Le modafinil est lГ©gГЁrement plus efficace le matin que le soir, et ne favorise pas la somnolence. Le modafinil est gГ©nГ©ralement disponible sous forme de comprimГ© de 200 mg. Le modafinil met un peu plus de temps Г  se dissoudre que les autres mГ©dicaments. Le modafinil peut ГЄtre utilisГ© pour traiter la narcolepsie et les troubles du sommeil liГ©s au travail postГ©. Le modafinil stimule efficacement ces centres "du sommeil", prГ©venant la somnolence lorsque l'on a besoin de se rГ©veiller et de gagner de l'Г©nergie. Le principal ingrГ©dient pharmaceutique actif du modafinil est le N-acГ©tyl-d-aspartyl-d-glutamate (NAAG), bien que la concentration exacte de cet ingrГ©dient ne soit pas connue. Il est approuvГ© aux Г‰tats-Unis pour traiter les troubles du sommeil liГ©s au travail postГ© ainsi que pour ГЄtre utilisГ© comme traitement d'appoint chez les personnes souffrant d'apnГ©e obstructive du sommeil.

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Le modafinil a un seuil thГ©rapeutique bas, avec des doses occasionnelles allant jusqu'Г  600 mg rapportГ©es. Les effets du modafinil sont similaires Г  ceux de l'amphГ©tamine ou de la cocaГЇne, mais la plupart des gens ne ressentent aucun de ses effets secondaires, tels que l'anxiГ©tГ©, l'agitation ou l'agitation. Ceci est rГ©alisГ© en bloquant le transporteur de dopamine prГ©synaptique. De plus, le modafinil est Г©tudiГ© pour voir s'il affecte la mГ©moire et les processus liГ©s Г  l'attention chez des volontaires sains et s'il peut amГ©liorer leur capacitГ© Г  effectuer des tГўches complexes. Le modafinil est disponible aux Г‰tats-Unis sous le nom de marque Provigil ou sous le nom commercial Alertec. L'administration concomitante de mГ©dicaments qui inhibent cette enzyme peut entraГ®ner une augmentation des concentrations du mГ©dicament. Le modafinil est mieux pris au petit-dГ©jeuner car il favorise la concentration et la vigilance. En tant que tel, 200 mg est devenu la dose la plus couramment utilisГ©e pour l'amГ©lioration cognitive. et Alertec. Il a Г©tГ© dГ©montrГ© que le modafinil a un effet puissant sur l'amГ©lioration des performances des sujets aux tests de mГ©moire lorsqu'il est pris tГґt dans la journГ©e. Cette Г©tude a conclu que la pГ©moline n'Г©tait pas un activateur cognitif efficace. Modafinil peut ГЄtre utilisГ© pour traiter les conditions mГ©dicales suivantes : Le modafinil peut Г©galement ГЄtre utilisГ© Г  des fins non rГ©pertoriГ©es dans ce guide de mГ©dicament. Le modafinil est transformГ© Г  partir d'un alcaloГЇde prГ©sent dans les feuilles de la plante mГ©dicinale vinca (Apocynaceae) appelГ©e apovincamine. Modafinil contient le composГ© chimique D-thrГ©o-3-mГ©thyl-2-pyrrolidinone. modiodal drogue Le modafinil semble agir en agissant sur la dopamine et en modulant les zones du cerveau impliquГ©es dans le cycle du sommeil. La nourriture ne semble pas affecter l'absorption ou le mГ©tabolisme du mГ©dicament. Il est Г©galement appelГ© Provigil, Generikum® Modafinil, Modalefenol et Modralift. Il est Г©galement disponible sur ordonnance en GrГЁce. C'est un stimulant non amphГ©tamine (un type de stimulant sans propriГ©tГ©s stimulantes). Ils sont gГ©nГ©ralement pris environ une heure avant le coucher. Le modafinil est un stimulant, mais ses effets pharmacologiques ne sont pas les mГЄmes que ceux de l'Г©phГ©dra. C'est la forme qui devient Г©ventuellement disponible pour la liaison avec les transporteurs de la dopamine et de la noradrГ©naline, ainsi qu'avec le transporteur de la sГ©rotonine. On pense Г©galement que des parties de l'hypothalamus latГ©ral, du raphГ© dorsal et du thalamus mГ©dial sont impliquГ©es. Le mГ©dicament modafinil est largement utilisГ© pour augmenter l'Г©veil, en particulier pour les professions dans lesquelles ils nГ©cessitent une concentration frГ©quente et soutenue Г  l'Г©tat de veille, bien qu'il puisse fonctionner pour les personnes qui ont gГ©nГ©ralement du mal Г  rester Г©veillГ©es pendant la journГ©e. La dose recommandГ©e de Modafinil pour la narcolepsie et d'autres troubles du sommeil est de 400 mg, quatre fois par jour. La posologie du modafinil dГ©pend de la condition traitГ©e.

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#8
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#9
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